Pimelic Diphenylamide 106
CAS No. 937039-45-7
Pimelic Diphenylamide 106 ( RGFA-8;TC-H 106;BRD-4657 )
产品货号. M16712 CAS No. 937039-45-7
A slow, tight-binding inhibitor of class I HDACs.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥340 | 有现货 |
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10MG | ¥543 | 有现货 |
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25MG | ¥932 | 有现货 |
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50MG | ¥1596 | 有现货 |
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100MG | ¥2908 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Pimelic Diphenylamide 106
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述A slow, tight-binding inhibitor of class I HDACs.
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产品描述A slow, tight-binding inhibitor of class I HDACs (HDAC1/2/3, Ki=148/102/14 nM respectively); shows weak inhibition on HDAC8 (IC50=5 uM); has preference toward HDAC3.
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同义词RGFA-8;TC-H 106;BRD-4657
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通路Cell Cycle/DNA Damage
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靶点HDAC
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受体HDAC
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研究领域Neurological Disease
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适应症——
化学信息
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CAS Number937039-45-7
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分子量339.43
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分子式C20H25N3O2
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 25 mg/mL
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SMILESO=C(NC1=CC=CC=C1N)CCCCCC(NC2=CC=C(C)C=C2)=O
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化学全称Heptanediamide, N1-(2-aminophenyl)-N7-(4-methylphenyl)-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Chou CJ, et al. J Biol Chem. 2008 Dec 19;283(51):35402-9.
2. Xu C, et al. Chem Biol. 2009 Sep 25;16(9):980-9.
2. Xu C, et al. Chem Biol. 2009 Sep 25;16(9):980-9.
产品手册
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